Prodrug Design

Written By Vivekkumar K Redasani
Prodrug Design
  • Publsiher : Academic Press
  • Release : 07 July 2015
  • ISBN : 0128035579
  • Pages : 84 pages
  • Rating : /5 from reviews
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Download or read book entitled Prodrug Design by author: Vivekkumar K Redasani which was release on 07 July 2015 and published by Academic Press with total page 84 pages . This book available in PDF, EPUB and Kindle Format. Prodrug Design: Perspectives, Approaches and Applications in Medicinal Chemistry provides a focused overview of this critical area of drug discovery, as that continuous process strives not only to discover new drug compounds but also to modify the existing ones. This valuable primer supports this mission of drug development and its goal of reducing undesired effects and improving therapeutic effectiveness of drug compounds. Providing a unique compilation of data, insightful case studies, and review of existing literature in the area, the book will promote innovation in medicinal and pharmaceutical chemistry research, exploring the limitations of existing drugs and their improvement. Prodrug Design reviews marketed compounds, the safety of promoieties, and a detailed classification of prodrugs organized by therapeutic area for easy reference. Offers unique, detailed overview of Prodrug research and literature Provides detailed chemical structures Includes Prodrug listing by therapeutic area

Prodrug Design

Prodrug Design
  • Author : Vivekkumar K Redasani,Sanjay B. Bari
  • Publisher : Academic Press
  • Release Date : 2015-07-07
  • Total pages : 84
  • ISBN : 0128035579
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Summary : Prodrug Design: Perspectives, Approaches and Applications in Medicinal Chemistry provides a focused overview of this critical area of drug discovery, as that continuous process strives not only to discover new drug compounds but also to modify the existing ones. This valuable primer supports this mission of drug development and its ...

Prodrugs Design

Prodrugs Design
  • Author : Rafik Karaman
  • Publisher : Nova Science Pub Incorporated
  • Release Date : 2014-07-01
  • Total pages : 277
  • ISBN : 0128035579
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Summary : The prodrug approach is a promising and well established strategy for the development of new entities that possess superior efficacy, selectivity and reduced toxicity. Hence an optimized therapeutic outcome can be accomplished using this approach. Prodrug design is becoming more elaborate in the development of efficient and selective drug delivery ...

Prodrugs and Targeted Delivery

Prodrugs and Targeted Delivery
  • Author : Jarkko Rautio
  • Publisher : John Wiley & Sons
  • Release Date : 2011-01-11
  • Total pages : 520
  • ISBN : 0128035579
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Summary : This topical reference and handbook addresses the chemistry, pharmacology, toxicology and the patentability of prodrugs, perfectly mirroring the integrated approach prevalent in today's drug design. It summarizes current experiences and strategies for the rational design of prodrugs, beginning at the early stages of the development process, as well as discussing ...

Drug Absorption Evaluation Prodrug Design and Intestinal Transporter Expression by Genechip Analysis

Drug Absorption Evaluation  Prodrug Design and Intestinal Transporter Expression by Genechip Analysis
  • Author : Duxin Sun
  • Publisher : Unknown
  • Release Date : 2002
  • Total pages : 212
  • ISBN : 0128035579
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Summary : Read online Drug Absorption Evaluation Prodrug Design and Intestinal Transporter Expression by Genechip Analysis written by Duxin Sun, published by which was released on 2002. Download full Drug Absorption Evaluation Prodrug Design and Intestinal Transporter Expression by Genechip Analysis Books now! Available in PDF, ePub and Kindle....

Design of Prodrugs

Design of Prodrugs
  • Author : Hans Bundgaard
  • Publisher : Elsevier Publishing Company
  • Release Date : 1985
  • Total pages : 360
  • ISBN : 0128035579
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Summary : Read online Design of Prodrugs written by Hans Bundgaard, published by Elsevier Publishing Company which was released on 1985. Download full Design of Prodrugs Books now! Available in PDF, ePub and Kindle....

Prodrug Designing of Nsaids

Prodrug Designing of Nsaids
  • Author : Smita Patil,Pramod Shirote,Rajendra Doijad
  • Publisher : LAP Lambert Academic Publishing
  • Release Date : 2012
  • Total pages : 104
  • ISBN : 0128035579
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Summary : Separation of therapeutic effects from toxicity is a valuable goal in the drug development process. Prodrug design is a part of the general drug discovery process, in which a unique combination of therapeutically active substances is observed to have desirable pharmacological effects. In human therapy prodrug designing has given successful ...

Development of Macromolecular Prodrug Conjugates for the Diagnosis and Treatment of Musculoskeletal Diseases

Development of Macromolecular Prodrug Conjugates for the Diagnosis and Treatment of Musculoskeletal Diseases
  • Author : Xin Wei
  • Publisher : Unknown
  • Release Date : 2018
  • Total pages : 206
  • ISBN : 0128035579
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Summary : Macromolecular prodrug conjugate is a promising strategy for better diagnosis and treatment of musculoskeletal diseases. Our lab has pioneered this effort and has successfully developed multiple prodrug formulations. The general approach we have taken is to incorporate active ingredient (AI, including imaging probe or therapeutic agents) containing monomers into water-soluble ...

Use of the Combination of Prodrug Design and Salt Optimization

Use of the Combination of Prodrug Design and Salt Optimization
  • Author : Anders Bach Nielsen
  • Publisher : Unknown
  • Release Date : 2004
  • Total pages : 82
  • ISBN : 0128035579
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Summary : Read online Use of the Combination of Prodrug Design and Salt Optimization written by Anders Bach Nielsen, published by which was released on 2004. Download full Use of the Combination of Prodrug Design and Salt Optimization Books now! Available in PDF, ePub and Kindle....

Recent Advancement in Prodrugs

Recent Advancement in Prodrugs
  • Author : Kamal Shah,Durgesh Nandini Chauhan,Nagendra Singh Chauhan,Pradeep Mishra
  • Publisher : CRC Press
  • Release Date : 2020-05-13
  • Total pages : 336
  • ISBN : 0128035579
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Summary : Recent Advancement in Prodrugs Drugs used as medicines have many limitations like low chemical stability, aqueous solubility, or oral absorption/bioavailability, rapid presystemic metabolism, toxicity, inadequate site specificity, or poor patient acceptance/compliance (unwanted adverse effects, unacceptable taste or odor, irritation or pain). Prodrugs design is an approach to overcome ...

Design Synthesis and Biological Evaluation of Glutathione Peptidomimetics as Components of Targeted Prodrugs and Glyoxalase 1 Inhibitors

Design  Synthesis and Biological Evaluation of Glutathione Peptidomimetics as Components of Targeted Prodrugs and Glyoxalase 1 Inhibitors
  • Author : Swati Sudhakar More
  • Publisher : Unknown
  • Release Date : 2007
  • Total pages : 434
  • ISBN : 0128035579
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Summary : Read online Design Synthesis and Biological Evaluation of Glutathione Peptidomimetics as Components of Targeted Prodrugs and Glyoxalase 1 Inhibitors written by Swati Sudhakar More, published by which was released on 2007. Download full Design Synthesis and Biological Evaluation of Glutathione Peptidomimetics as Components of Targeted Prodrugs and Glyoxalase 1 Inhibitors Books now! Available ...

Hydrolysis in Drug and Prodrug Metabolism

Hydrolysis in Drug and Prodrug Metabolism
  • Author : Bernard Testa,Joachim M. Mayer,Joachim Mayer
  • Publisher : John Wiley & Sons
  • Release Date : 2003-08
  • Total pages : 780
  • ISBN : 0128035579
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Summary : Many drugs and other xenobiotics (e.g., preservatives, insecticides, and plastifiers) contain hydrolyzable moieties such as ester or amide groups. In biological media, such foreign compounds are, therefore, important substrates for hydrolytic reactions catalyzed by hydrolases or proceeding non-enzymatically. Despite their significance, until now, no book has been dedicated to ...

Optimisation of Solubility Parameter and Enzyme Specificity in Haloperidol Prodrug Design

Optimisation of Solubility Parameter and Enzyme Specificity in Haloperidol Prodrug Design
  • Author : Andrew Morris
  • Publisher : Unknown
  • Release Date : 2003
  • Total pages : 490
  • ISBN : 0128035579
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Summary : Read online Optimisation of Solubility Parameter and Enzyme Specificity in Haloperidol Prodrug Design written by Andrew Morris, published by which was released on 2003. Download full Optimisation of Solubility Parameter and Enzyme Specificity in Haloperidol Prodrug Design Books now! Available in PDF, ePub and Kindle....

Drug Design

Drug Design
  • Author : Georges Jolles,K. R. H. Wooldridge
  • Publisher : Unknown
  • Release Date : 1984
  • Total pages : 268
  • ISBN : 0128035579
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Summary : Ovulation/implan...

Textbook of Drug Design and Discovery Third Edition

Textbook of Drug Design and Discovery  Third Edition
  • Author : Tommy Liljefors,Povl Krogsgaard-Larsen,Ulf Madsen
  • Publisher : CRC Press
  • Release Date : 2002-07-25
  • Total pages : 592
  • ISBN : 0128035579
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Summary : Building on the success of the previous editions, Textbook of Drug Design and Discovery has been thoroughly revised and updated to provide a complete source of information on all facets of drug design and discovery for students of chemistry, pharmacy, pharmacology, biochemistry, and medicine. The book follows drug design from ...

Drug Discovery Handbook

Drug Discovery Handbook
  • Author : Shayne Cox Gad
  • Publisher : John Wiley & Sons
  • Release Date : 2005-07-08
  • Total pages : 1496
  • ISBN : 0128035579
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Summary : The Drug Discovery Handbook gives professionals a tool tofacilitate drug discovery by bringing together, for the first timein one resource, a compendium of methods and techniques that needto be considered when developing new drugs. This comprehensive, practical guide presents an explanation of thelatest techniques and methods in drug discovery, including: ...