Oligomerization and Allosteric Modulation in G Protein Coupled Receptors

Written By Anonim
Oligomerization and Allosteric Modulation in G Protein Coupled Receptors
  • Publsiher : Academic Press
  • Release : 02 December 2012
  • ISBN : 012394791X
  • Pages : 488 pages
  • Rating : /5 from reviews
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Download or read book entitled Oligomerization and Allosteric Modulation in G Protein Coupled Receptors by author: Anonim which was release on 02 December 2012 and published by Academic Press with total page 488 pages . This book available in PDF, EPUB and Kindle Format. In this thematic volume of Progress in Molecular Biology and Translational Science, researchers reflect on recent developments and research surrounding G protein-coupled receptors. The chapters cover a large breadth of research, including GPCR role in stem cell function and pharmacology. Authors explore in-depth research techniques and applications of GPCR usage, covering theory, laboratory approaches, and unique qualities that make GPCRs a crucial tool in microbiological and cancer research. Contributions from leading authorities Informs and updates on all the latest developments in the field

Oligomerization and Allosteric Modulation in G Protein Coupled Receptors

Oligomerization and Allosteric Modulation in G Protein Coupled Receptors
  • Author : Anonim
  • Publisher : Academic Press
  • Release Date : 2012-12-02
  • Total pages : 488
  • ISBN : 012394791X
GET BOOK

Summary : In this thematic volume of Progress in Molecular Biology and Translational Science, researchers reflect on recent developments and research surrounding G protein-coupled receptors. The chapters cover a large breadth of research, including GPCR role in stem cell function and pharmacology. Authors explore in-depth research techniques and applications of GPCR usage, ...

From Structure to Clinical Development Allosteric Modulation of G Protein Coupled Receptors

From Structure to Clinical Development  Allosteric Modulation of G Protein Coupled Receptors
  • Author : Anonim
  • Publisher : Academic Press
  • Release Date : 2020-05-13
  • Total pages : 328
  • ISBN : 012394791X
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Summary : From Structure to Clinical Development: Allosteric Modulation of G Protein-Coupled Receptors, Volume 88, the latest release in the Advances in Pharmacology series, presents a variety of chapters from the best authors in the field. Chapters in this updated edition include Targeting muscarinic M1 receptor in neurodegeneration, Photo‐switchable allosteric ligands, Computational ...

Allosteric Modulation of G Protein coupled Receptors

Allosteric Modulation of G Protein coupled Receptors
  • Author : Lauren Therese May
  • Publisher : Unknown
  • Release Date : 2007
  • Total pages : 430
  • ISBN : 012394791X
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Summary : Read online Allosteric Modulation of G Protein coupled Receptors written by Lauren Therese May, published by which was released on 2007. Download full Allosteric Modulation of G Protein coupled Receptors Books now! Available in PDF, ePub and Kindle....

Allosteric Modulation of G Protein coupled Receptors

Allosteric Modulation of G Protein coupled Receptors
  • Author : Joaquin Botta
  • Publisher : Unknown
  • Release Date : 2018
  • Total pages : 212
  • ISBN : 012394791X
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Summary : Read online Allosteric Modulation of G Protein coupled Receptors written by Joaquin Botta, published by which was released on 2018. Download full Allosteric Modulation of G Protein coupled Receptors Books now! Available in PDF, ePub and Kindle....

Allosteric Modulation of G Protein coupled Receptors

Allosteric Modulation of G Protein coupled Receptors
  • Author : Zhan-Guo Gao
  • Publisher : Unknown
  • Release Date : 2000
  • Total pages : 188
  • ISBN : 012394791X
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Summary : Read online Allosteric Modulation of G Protein coupled Receptors written by Zhan-Guo Gao, published by which was released on 2000. Download full Allosteric Modulation of G Protein coupled Receptors Books now! Available in PDF, ePub and Kindle....

Allosteric Modulation by Sodium Ions and Amilorides of G Protein coupled Receptors

Allosteric Modulation by Sodium Ions and Amilorides of G Protein coupled Receptors
  • Author : Anonim
  • Publisher : Unknown
  • Release Date : 2016
  • Total pages : 181
  • ISBN : 012394791X
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Summary : Read online Allosteric Modulation by Sodium Ions and Amilorides of G Protein coupled Receptors written by , published by which was released on 2016. Download full Allosteric Modulation by Sodium Ions and Amilorides of G Protein coupled Receptors Books now! Available in PDF, ePub and Kindle....

Protein Allostery in Drug Discovery

Protein Allostery in Drug Discovery
  • Author : Jian Zhang,Ruth Nussinov
  • Publisher : Springer Nature
  • Release Date : 2019-11-09
  • Total pages : 384
  • ISBN : 012394791X
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Summary : The book focuses on protein allostery in drug discovery. Allosteric regulation, ʹthe second secret of lifeʹ, fine-tunes virtually most biological processes and controls physiological activities. Allostery can both cause human diseases and contribute to development of new therapeutics. Allosteric drugs exhibit unparalleled advantages compared to conventional orthosteric drugs, rendering the ...

Allosteric Receptor Modulation in Drug Targeting

Allosteric Receptor Modulation in Drug Targeting
  • Author : Norman G. Bowery
  • Publisher : CRC Press
  • Release Date : 2016-04-19
  • Total pages : 376
  • ISBN : 012394791X
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Summary : Offering a wide array of illustrations and tables in every chapter, this book extensively covers the principles of allosterism in reference to drug action and progresses to a detailed examination of individual ionotropic and G-protein coupled receptor systems-helping those new to the subject understand the importance of allosterism and providing ...

Biased Signaling and Allosteric Modulation of the Angiotensin II Type 1 Receptor

Biased Signaling and Allosteric Modulation of the Angiotensin II Type 1 Receptor
  • Author : Stephanie Clement
  • Publisher : Unknown
  • Release Date : 2016
  • Total pages : 212
  • ISBN : 012394791X
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Summary : "G protein coupled receptors (GPCR) represent over 30% of drug targets and are involved in nearly all physiological and cellular responses. The angiotensin II (AngII) type I receptor (AT1R) is an important member of this receptor family. Its main endogenous ligand is the hormone angiotensin II (AngII), which regulates blood ...

Dimer dependent Allosteric Modulation Within GPCR Signalling Complexes Can Influence Signalling Diversity

Dimer dependent Allosteric Modulation Within GPCR Signalling Complexes Can Influence Signalling Diversity
  • Author : Katrin Altosaar
  • Publisher : Unknown
  • Release Date : 2013
  • Total pages : 212
  • ISBN : 012394791X
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Summary : "G protein-coupled receptors (GPCRs) comprise the largest group of cell surface receptors, translating environmental signals into cellular responses via cognate G protein partners. Contrary to our initial understanding, most GPCRs do not function in living cells as monomers, but most likely dimers, or even larger arrays of receptors. Standard drug ...

Allosteric Modulation of the CB1 Receptor

Allosteric Modulation of the CB1 Receptor
  • Author : Jamie Kerr
  • Publisher : Unknown
  • Release Date : 2013
  • Total pages : 212
  • ISBN : 012394791X
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Summary : Bioactive compounds from Cannabis sativa have been used for millennia to alleviate the symptoms of a range of diseases. The physiological basis of effects such as analgesia, stimulation of hunger and reduction of inflammation was established in the late 20th century with the discovery of cannabinoid receptors but efforts to ...

Pharmacology of G Protein Coupled Receptors

Pharmacology of G Protein Coupled Receptors
  • Author : S. J. Enna
  • Publisher : Academic Press
  • Release Date : 2011
  • Total pages : 391
  • ISBN : 012394791X
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Summary : G protein coupled receptors remain the most important class of therapeutic targets in medicine. In the last 5 years, tremendous advances have been made in our understanding of the structure and mechanism of this critical family of drug targets. The present volume explores the modern experimental and conceptual framework for drug ...

Exploring Aspects of Allosteric Modulation and Bias Signalling at the Glucagon like Peptide 1 Receptor

Exploring Aspects of Allosteric Modulation and Bias Signalling at the Glucagon like Peptide 1 Receptor
  • Author : Emilia Elizabeth Savage
  • Publisher : Unknown
  • Release Date : 2015
  • Total pages : 544
  • ISBN : 012394791X
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Summary : The glucagon-like peptide-1 receptor (GLP-1R) is an important regulator of insulin biosynthesis and secretion, and is one of the key therapeutic targets in the management of type II diabetes mellitus and obesity. Like most GPCRs, the GLP-1R is pleiotropically coupled, to physiologically relevant signalling pathways including cAMP formation, ...

G Protein Coupled Receptors in Drug Discovery

G Protein Coupled Receptors in Drug Discovery
  • Author : Marta Filizola
  • Publisher : Humana Press
  • Release Date : 2018-02-21
  • Total pages : 327
  • ISBN : 012394791X
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Summary : This detailed volume provides an overview of recent techniques employed in the field of G protein-coupled receptors (GPCRs) to screen for new drugs and to derive information about their receptor structure, dynamics, and function for the purpose of developing improved therapeutics. Owing to remarkable recent advances in the structural, biophysical ...

Allosteric Modulators of Serotonin and Dopamine Receptors

Allosteric Modulators of Serotonin and Dopamine Receptors
  • Author : Javier García Cárceles
  • Publisher : Unknown
  • Release Date : 2017
  • Total pages : 220
  • ISBN : 012394791X
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Summary : G protein-coupled receptors (GPCRs) are eukaryotic cell membrane proteins that transduce a wide range of extracellular stimuli into intracellular changes in cell function. Based on their amino acid sequence, they can be classified in four different classes: class A or rhodopsin-like family, class B or secretin-like family, class C or ...